Novel b-raf inhibitors devoid of rapid metabolism and of binding to pregnane x receptor

The present invention relates to N-(3-(5-(pyrimidin-4-yl)thiazol-4-yl)phenylsulfonamide compounds which are useful as inhibitors of protein kinases, more specifically BRAF or mutant forms thereof, to pharmaceutical composition comprising such compounds, and to uses of such compounds in the treatment or prevention of diseases associated with deregulated protein kinase activity, such as cancer.

Keywords: BRAF inhibitors
Patent Application number: European Procedure (Patents) (EPA) - 05 Déc. 2019 - 19 306 579.4
Inventors:
LABESSE GillesCOHEN-GONSAUD MartinBOURGUET WilliamGELIN MurielGUICHOU Jean-FrançoisBALAGUER PatrickSCHNEIDER Mélanie
Publications:
null

Reference:

CHIM18530-T1

    Business Developper
    contact
    Aymeric Empereur
    Business Developer
    Patent filling date: 05-12-2019
    Rare disease: No
    Second indication: No

    You might also be interested in